Total synthesis of dapiramicin B

Hiroyuki Ohno, Takashi Terui, Takafumi Kitawaki, Noritaka Chida

Research output: Contribution to journalArticlepeer-review

9 Citations (Scopus)


The first total synthesis of dapiramicin B, a nucleoside antibiotic, is described. The characteristic N-glycoside linkage in dapiramicin B was effectively constructed by way of the Pd-catalyzed coupling reaction of a heptopyranosylamine with a bromopyrrolopyrimidine derivative.

Original languageEnglish
Pages (from-to)5747-5750
Number of pages4
JournalTetrahedron Letters
Issue number32
Publication statusPublished - 2006 Aug 7


  • Dapiramicin B
  • N-Arylation
  • Nucleoside antibiotic
  • Pd-Catalyzed
  • Total synthesis

ASJC Scopus subject areas

  • Biochemistry
  • Drug Discovery
  • Organic Chemistry


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