抄録
Preparation of N-alkylated 2-epi-valienamines was accomplished by the palladium-catalyzed coupling reaction of the allylic chloride 5 with various amines in the presence of trimethylolpropane phosphite (TMPP). The 2-epi-valienamine precursor (i.e. allylic chloride 5) was obtained from the reaction of diol 2 with Viehe's salt and the diol 2 was readily prepared from (-)-quinic acid in 10 steps. (C) 2000 Elsevier Science Ltd.
| 本文言語 | English |
|---|---|
| ページ（範囲） | 6865-6868 |
| ページ数 | 4 |
| ジャーナル | Tetrahedron Letters |
| 巻 | 41 |
| 号 | 35 |
| DOI | |
| 出版ステータス | Published - 2000 8 26 |
ASJC Scopus subject areas
- Biochemistry
- Drug Discovery
- Organic Chemistry