抄録
Preparation of N-alkylated 2-epi-valienamines was accomplished by the palladium-catalyzed coupling reaction of the allylic chloride 5 with various amines in the presence of trimethylolpropane phosphite (TMPP). The 2-epi-valienamine precursor (i.e. allylic chloride 5) was obtained from the reaction of diol 2 with Viehe's salt and the diol 2 was readily prepared from (-)-quinic acid in 10 steps. (C) 2000 Elsevier Science Ltd.
本文言語 | English |
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ページ(範囲) | 6865-6868 |
ページ数 | 4 |
ジャーナル | Tetrahedron Letters |
巻 | 41 |
号 | 35 |
DOI | |
出版ステータス | Published - 2000 8月 26 |
ASJC Scopus subject areas
- 生化学
- 創薬
- 有機化学