Total synthesis of dapiramicin B

Hiroyuki Ohno, Takashi Terui, Takafumi Kitawaki, Noritaka Chida

研究成果: Article

8 引用 (Scopus)

抄録

The first total synthesis of dapiramicin B, a nucleoside antibiotic, is described. The characteristic N-glycoside linkage in dapiramicin B was effectively constructed by way of the Pd-catalyzed coupling reaction of a heptopyranosylamine with a bromopyrrolopyrimidine derivative.

元の言語English
ページ(範囲)5747-5750
ページ数4
ジャーナルTetrahedron Letters
47
発行部数32
DOI
出版物ステータスPublished - 2006 8 7

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Glycosides
Nucleosides
Anti-Bacterial Agents
Derivatives
dapiramicin B

ASJC Scopus subject areas

  • Biochemistry
  • Organic Chemistry
  • Drug Discovery

これを引用

Total synthesis of dapiramicin B. / Ohno, Hiroyuki; Terui, Takashi; Kitawaki, Takafumi; Chida, Noritaka.

:: Tetrahedron Letters, 巻 47, 番号 32, 07.08.2006, p. 5747-5750.

研究成果: Article

Ohno, H, Terui, T, Kitawaki, T & Chida, N 2006, 'Total synthesis of dapiramicin B', Tetrahedron Letters, 巻. 47, 番号 32, pp. 5747-5750. https://doi.org/10.1016/j.tetlet.2006.06.001
Ohno, Hiroyuki ; Terui, Takashi ; Kitawaki, Takafumi ; Chida, Noritaka. / Total synthesis of dapiramicin B. :: Tetrahedron Letters. 2006 ; 巻 47, 番号 32. pp. 5747-5750.
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